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Binding Mode Characterization of NBD Series CD4-Mimetic HIV-1 Entry Inhibitors by X-Ray Structure and Resistance Study

We previously identified two small-molecule CD4 mimetics—NBD-556 and NBD-557—and synthesized a series of NBD compounds that resulted in improved neutralization activity in a single-cycle HIV-1 infectivity assay. For the current investigation, we selected several of the most active compounds and asse...

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Autores principales: Curreli, Francesca, Kwon, Young Do, Zhang, Hongtao, Yang, Yongping, Scacalossi, Daniel, Kwong, Peter D., Debnath, Asim K.
Formato: Artigo
Lenguaje:Inglês
Publicado: American Society for Microbiology 2014
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC4135886/
https://ncbi.nlm.nih.gov/pubmed/25001301
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.03339-14
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