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N-Boc Amines to Oxazolidinones via Pd(II)/Bis-sulfoxide/Brønsted Acid Co-Catalyzed Allylic C–H Oxidation

[Image: see text] A Pd(II)/bis-sulfoxide/Brønsted acid catalyzed allylic C–H oxidation reaction for the synthesis of oxazolidinones from simple N-Boc amines is reported. A range of oxazolidinones are furnished in good yields (avg 63%) and excellent diastereoselectivities (avg 15:1) to furnish produc...

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Detalhes bibliográficos
Main Authors: Osberger, Thomas J., White, M. Christina
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2014
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4132963/
https://ncbi.nlm.nih.gov/pubmed/24999765
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja506036q
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