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Using ‘biased-privileged’ scaffolds to identify lysine methyltransferase inhibitors

Methylation of histones by lysine methyltransferases (KMTases) plays important roles in regulating chromatin function. It is also now clear that improper KMTases activity is linked to human diseases, such as cancer. We report an approach that employs drug-like ‘privileged’ scaffolds biased with moti...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Kashyap, Sudhir, Sandler, Joel, Martinez, Eduardo J., Kapoor, Tarun M.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2014
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC4038709/
https://ncbi.nlm.nih.gov/pubmed/24650704
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2014.02.024
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