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Using ‘biased-privileged’ scaffolds to identify lysine methyltransferase inhibitors

Methylation of histones by lysine methyltransferases (KMTases) plays important roles in regulating chromatin function. It is also now clear that improper KMTases activity is linked to human diseases, such as cancer. We report an approach that employs drug-like ‘privileged’ scaffolds biased with moti...

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Bibliografski detalji
Glavni autori: Kashyap, Sudhir, Sandler, Joel, Martinez, Eduardo J., Kapoor, Tarun M.
Format: Artigo
Jezik:Inglês
Izdano: 2014
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4038709/
https://ncbi.nlm.nih.gov/pubmed/24650704
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2014.02.024
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