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Designing bifunctional NOP receptor-mu opioid receptor ligands from NOP-receptor selective scaffolds. Part II

The nociceptin opioid receptor (NOP) and its endogenous peptide ligand nociceptin/orphanin FQ have been shown to modulate the pharmacological effects of the classical opioid receptor system. Suppression of opioid-induced reward associated with mu-opioid receptor (MOP)-mediated analgesia, without dec...

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Autores principales: Journigan, V. Blair, Polgar, Willma, Khroyan, Taline V., Zaveri, Nurulain T.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2014
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC4033624/
https://ncbi.nlm.nih.gov/pubmed/24657054
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2014.02.047
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