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Evaluation and Structural Basis for the Inhibition of Tankyrases by PARP Inhibitors

[Image: see text] Tankyrases, an enzyme subfamily of human poly(ADP-ribosyl)polymerases, are potential drug targets especially against cancer. We have evaluated inhibition of tankyrases by known PARP inhibitors and report five cocrystal structures of the most potent compounds in complex with human t...

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Bibliografiske detaljer
Main Authors: Haikarainen, Teemu, Narwal, Mohit, Joensuu, Päivi, Lehtiö, Lari
Format: Artigo
Sprog:Inglês
Udgivet: American Chemical Society 2013
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4027629/
https://ncbi.nlm.nih.gov/pubmed/24900770
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml400292s
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