A carregar...

Structural Basis for Potency and Promiscuity in Poly(ADP-ribose) Polymerase (PARP) and Tankyrase Inhibitors

Selective inhibitors could help unveil the mechanisms by which inhibition of poly(ADP-ribose) polymerases (PARPs) elicits clinical benefits in cancer therapy. We profiled 10 clinical PARP inhibitors and commonly used research tools for their inhibition of multiple PARP enzymes. We also determined cr...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Thorsell, Ann-Gerd, Ekblad, Torun, Karlberg, Tobias, Löw, Mirjam, Pinto, Ana Filipa, Trésaugues, Lionel, Moche, Martin, Cohen, Michael S., Schüler, Herwig
Formato: Artigo
Idioma:Inglês
Publicado em: 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5934274/
https://ncbi.nlm.nih.gov/pubmed/28001384
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.6b00990
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!