Загрузка...

Analysis of Flexibility and Hotspots in Bcl-xL and Mcl-1 Proteins for the Design of Selective Small-Molecule Inhibitors

[Image: see text] Although Bcl-xL and Mcl-1, two antideath Bcl-2 members, have similar, flexible binding sites, they can achieve high binding selectivity to endogenous binding partners and synthetic small-molecule inhibitors. Here, we employed molecular dynamic (MD) simulations and hotspot analysis...

Полное описание

Сохранить в:
Библиографические подробности
Главные авторы: Yang, Chao-Yie, Wang, Shaomeng
Формат: Artigo
Язык:Inglês
Опубликовано: American Chemical Society 2012
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC4025761/
https://ncbi.nlm.nih.gov/pubmed/24900469
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml200301w
Метки: Добавить метку
Нет меток, Требуется 1-ая метка записи!