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Targeting MUC1-C is synergistic with bortezomib in downregulating TIGAR and inducing ROS-mediated myeloma cell death

The proteosome inhibitor bortezomib (BTZ) induces endoplasmic reticulum and oxidative stress in multiple myeloma (MM) cells. The mucin 1 C-terminal subunit (MUC1-C) oncoprotein is aberrantly expressed in most MM cells, and targeting MUC1-C with GO-203, a cell-penetrating peptide inhibitor of MUC1-C...

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Detaylı Bibliyografya
Asıl Yazarlar: Yin, Li, Kufe, Turner, Avigan, David, Kufe, Donald
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: American Society of Hematology 2014
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC4014842/
https://ncbi.nlm.nih.gov/pubmed/24632713
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1182/blood-2013-11-539395
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