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‘Null Method’ Determination of Drug Biophase Concentration

PK/PD modeling is enhanced by improvements in the accuracy of its metrics. For PK/PD modeling of drugs and biologics that interact with enzymes or receptors, the equilibrium constant of the interaction can provide critical insight. Methodologies such as radioliogand binding and isolated tissue prepa...

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Autors principals: Tallarida, Ronald J., Lamarre, Neil, Raffa, Robert B.
Format: Artigo
Idioma:Inglês
Publicat: 2011
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4005008/
https://ncbi.nlm.nih.gov/pubmed/22037914
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11095-011-0612-5
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