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Identifying Barbiturate Binding Sites in a Nicotinic Acetylcholine Receptor with [(3)H]Allyl m-Trifluoromethyldiazirine Mephobarbital, a Photoreactive Barbiturate

At concentrations that produce anesthesia, many barbituric acid derivatives act as positive allosteric modulators of inhibitory GABA(A) receptors (GABA(A)Rs) and inhibitors of excitatory nicotinic acetylcholine receptors (nAChRs). Recent research on [(3)H]R-mTFD-MPAB ([(3)H]R-5-allyl-1-methyl-5-(m-t...

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Dettagli Bibliografici
Autori principali: Hamouda, Ayman K., Stewart, Deirdre S., Chiara, David C., Savechenkov, Pavel Y., Bruzik, Karol S., Cohen, Jonathan B.
Natura: Artigo
Lingua:Inglês
Pubblicazione: The American Society for Pharmacology and Experimental Therapeutics 2014
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3990015/
https://ncbi.nlm.nih.gov/pubmed/24563544
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.113.090985
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