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Selective ALDH3A1 Inhibition by Benzimidazole Analogues Increase Mafosfamide Sensitivity in Cancer Cells

[Image: see text] Aldehyde dehydrogenase enzymes irreversibly oxidize aldehydes generated from metabolism of amino acids, fatty acids, food, smoke, additives, and xenobiotic drugs. Cyclophosphamide is one such xenobiotic used in cancer therapies. Upon activation, cyclophosphamide forms an intermedia...

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Detalhes bibliográficos
Main Authors: Parajuli, Bibek, Fishel, Melissa L., Hurley, Thomas D.
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2014
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3988914/
https://ncbi.nlm.nih.gov/pubmed/24387105
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm401508p
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