Wird geladen...

Novel Histone Deacetylase Inhibitors with Enhanced Enzymatic Inhibition Effects and Potent in vitro and in vivo Anti-tumor Activities

In the present work, a series of small molecules were designed and synthesized based on structural optimization. Significant improvement in the enzymatic inhibition activity of the synthesized compounds was discovered. Moreover, tested compounds have moderate preference for class I HDACs over HDAC6...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: Zhang, Lei, Zhang, Yingjie, Chou, C. James, Inks, Elizabeth S., Wang, Xuejian, Li, Xiaoguang, Hou, Jinning, Xu, Wenfang
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2013
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3947464/
https://ncbi.nlm.nih.gov/pubmed/24227760
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.201300297
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!