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Conjugation of Vitamin E Analog α-TOS to Pt(IV) Complexes for Dual-Targeting Anticancer Therapy

We report two platinum(IV) complexes conjugated with a vitamin E analog, α-tocopherol succinate (α-TOS). One of the conjugates displays the activity of both cisplatin and αTOS in cancer cells, causing damage to DNA and mitochondria simultaneously. Accordingly, it serves as promising dual-targeting a...

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Autors principals: Suntharalingam, Kogularamanan, Song, Ying, Lippard, Stephen J.
Format: Artigo
Idioma:Inglês
Publicat: 2014
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3938893/
https://ncbi.nlm.nih.gov/pubmed/24452361
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c3cc48740g
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