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Combination Small Molecule MEK and PI3K Inhibition Enhances Uveal Melanoma Cell Death in a Mutant GNAQ and GNA11 Dependent Manner

PURPOSE: Activating Q209L/P mutations in GNAQ or GNA11 (GNAQ/11) are present in ∼ 80% of uveal melanomas (UM). Mutant GNAQ/11 are not currently therapeutically targetable. Inhibiting key downstream effectors of GNAQ/11 represents a rational therapeutic approach for UMs that harbor these mutations. T...

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Detalles Bibliográficos
Main Authors: Khalili, Jahan S., Yu, Xiaoxing, Wang, Ji, Hayes, Brendan C., Davies, Michael A., Lizee, Gregory, Esmaeli, Bita, Woodman, Scott E.
Formato: Artigo
Idioma:Inglês
Publicado: 2012
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC3935730/
https://ncbi.nlm.nih.gov/pubmed/22733540
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1078-0432.CCR-11-3227
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