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MLS-2384, a new 6-bromoindirubin derivative with dual JAK/Src kinase inhibitory activity, suppresses growth of diverse cancer cells

Janus kinase (JAK) and Src kinase are the two major tyrosine kinase families upstream of signal transducer and activator of transcription (STAT). Among the seven STAT family proteins, STAT3 is constitutively activated in many diverse cancers. Upon activation, JAK and Src kinases phosphorylate STAT3,...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Päätekijät: Liu, Lucy, Gaboriaud, Nicolas, Vougogianopoulou, Konstantina, Tian, Yan, Wu, Jun, Wen, Wei, Skaltsounis, Leandros, Jove, Richard
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: Landes Bioscience 2014
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC3928133/
https://ncbi.nlm.nih.gov/pubmed/24100507
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.4161/cbt.26721
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