A carregar...

Synthesis and evaluation of 4-substituted piperidines and piperazines as balanced affinity µ opioid receptor (MOR) agonist/δ opioid receptor (DOR) antagonist ligands

In this report, we describe a series of 4-substituted piperidine and piperazine compounds based on tetrahydroquinoline 1, a compound that shows balanced, low nanomolar binding affinity for the mu opioid receptor (MOR) and the delta opioid receptor (DOR). We have shown that by changing the length and...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Main Authors: Bender, Aaron M., Clark, Mary J., Agius, Michael P., Traynor, John R., Mosberg, Henry I.
Formato: Artigo
Idioma:Inglês
Publicado em: 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3919453/
https://ncbi.nlm.nih.gov/pubmed/24365161
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2013.12.021
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!