Wird geladen...

Inverse agonism of histamine H2 antagonist accounts for upregulation of spontaneously active histamine H2 receptors.

Histamine H2 receptors transfected in Chinese hamster ovary (CHO) cells are time- and dose-dependently upregulated upon exposure to the H2 antagonists cimetidine and ranitidine. This effect appears to be H2 receptor-mediated as no change in receptor density was observed after H1 or H3 antagonist tre...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: Smit, M J, Leurs, R, Alewijnse, A E, Blauw, J, Van Nieuw Amerongen, G P, Van De Vrede, Y, Roovers, E, Timmerman, H
Format: Artigo
Sprache:Inglês
Veröffentlicht: 1996
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC39108/
https://ncbi.nlm.nih.gov/pubmed/8692899
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!