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Reverse Yeast Two-hybrid System to Identify Mammalian Nuclear Receptor Residues that Interact with Ligands and/or Antagonists

As a critical regulator of drug metabolism and inflammation, Pregnane X Receptor (PXR), plays an important role in disease pathophysiology linking metabolism and inflammation (e.g. hepatic steatosis)(1,2). There has been much progress in the identification of agonist ligands for PXR, however, there...

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Autors principals: Li, Hao, Dou, Wei, Padikkala, Emil, Mani, Sridhar
Format: Artigo
Idioma:Inglês
Publicat: MyJove Corporation 2013
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3904218/
https://ncbi.nlm.nih.gov/pubmed/24300333
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3791/51085
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