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Reverse Yeast Two-hybrid System to Identify Mammalian Nuclear Receptor Residues that Interact with Ligands and/or Antagonists

As a critical regulator of drug metabolism and inflammation, Pregnane X Receptor (PXR), plays an important role in disease pathophysiology linking metabolism and inflammation (e.g. hepatic steatosis)(1,2). There has been much progress in the identification of agonist ligands for PXR, however, there...

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Detalhes bibliográficos
Main Authors: Li, Hao, Dou, Wei, Padikkala, Emil, Mani, Sridhar
Formato: Artigo
Idioma:Inglês
Publicado em: MyJove Corporation 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3904218/
https://ncbi.nlm.nih.gov/pubmed/24300333
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3791/51085
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