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Dopamine D3 Receptor Selective Ligands with Varying Intrinsic Efficacies at Adenylyl Cyclase Inhibition and Mitogenic Signaling Pathways

A panel of eight structurally related pairs of 2,3-dichloro and 2-methoxy substituted 4-phenylpiperazines with nanomolar affinity and selectivity at D3 dopamine receptors has been synthesized. Compounds in which a heterocyclic (2-phenyl pyridyl, 3-phenyl pyridyl, benzothiophen or benzofuran) moiety...

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Библиографические подробности
Главные авторы: Taylor, Michelle, Grundt, Peter, Griffin, Suzy A., Newman, Amy Hauck, Luedtke, Robert R.
Формат: Artigo
Язык:Inglês
Опубликовано: 2010
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC3821045/
https://ncbi.nlm.nih.gov/pubmed/19924694
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/syn.20725
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