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Synthesis of Sequence-Specific DNA-Protein Conjugates via a Reductive Amination Strategy

DNA-protein cross-links (DPCs) are ubiquitous, structurally diverse DNA lesions formed upon exposure to bis-electrophiles, transition metals, UV light, and reactive oxygen species. Because of their super-bulky, helix distorting nature, DPCs interfere with DNA replication, transcription, and repair,...

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Autores principales: Wickramaratne, Susith, Mukherjee, Shivam, Villalta, Peter W., Schärer, Orlando D., Tretyakova, Natalia
Formato: Artigo
Lenguaje:Inglês
Publicado: 2013
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3799944/
https://ncbi.nlm.nih.gov/pubmed/23885807
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bc400018u
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