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N,C-capped dipeptides with selectivity for mycobacterial proteasome over human proteasomes: Role of S3 and S1 binding pockets

We identified N,C-capped dipeptides that are selective for the Mycobacterium tuberculosis proteasome over human constitutive and immunoproteasomes. Differences in S3 and S1 binding pockets appeared to account for species-selectivity. The inhibitors are able to penetrate mycobacteria and kill non-rep...

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Detalhes bibliográficos
Main Authors: Lin, Gang, Chidawanyika, Tamutenda, Tsu, Christopher, Warrier, Thulasi, Vaubourgeix, Julien, Blackburn, Christopher, Gigstad, Kenneth, Sintchak, Michael, Dick, Lawrence, Nathan, Carl
Formato: Artigo
Idioma:Inglês
Publicado em: 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3773049/
https://ncbi.nlm.nih.gov/pubmed/23782398
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja400021x
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