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Total Synthesis of (+)-Trienomycins A and F via C-C Bond-Forming Hydrogenation and Transfer Hydrogenation

The triene-containing C17-benzene ansamycins trienomycins A and F are prepared in 16 steps (longest linear sequence, LLS) and 28 total steps. The C11-C13 stereotriad is prepared via enantioselective ruthenium catalyzed alcohol CH-syn-crotylation followed by chelation-controlled carbonyl dienylation....

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Del Valle, David J., Krische, Michael J.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2013
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC3757526/
https://ncbi.nlm.nih.gov/pubmed/23862627
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja4061273
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