A carregar...

Conformationally constrained analogs of BAY 59–3074 as novel cannabinoid receptor ligands

To obtain information on the pharmacophoric requirements of the CB1/CB2 partial agonist BAY 59–3074 we have synthesized a series of new conformationally constrained dibenzofuran (4a–d) and dibenzopyran analogs (5). All constrained analogs exhibited reduced binding affinity at both cannabinoid recept...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Main Authors: Teng, Heidi, Thakur, Ganesh A., Makriyannis, Alexandros
Formato: Artigo
Idioma:Inglês
Publicado em: 2011
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3693451/
https://ncbi.nlm.nih.gov/pubmed/21880487
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2011.07.017
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!