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A Perfluoroaryl-Cysteine S(N)Ar Chemistry Approach to Unprotected Peptide Stapling

We report the discovery of a facile transformation between perfluoroaromatic molecules and a cysteine thiolate, which is arylated at room temperature. This new approach enabled us to selectively modify cysteine residues in unprotected peptides, providing access to variants containing rigid perfluoro...

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Autors principals: Spokoyny, Alexander M., Zou, Yekui, Ling, Jingjing J., Yu, Hongtao, Lin, Yu-Shan, Pentelute, Bradley L.
Format: Artigo
Idioma:Inglês
Publicat: 2013
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3675880/
https://ncbi.nlm.nih.gov/pubmed/23560559
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja400119t
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