Loading...

Enantioselective synthesis of (R)-tolterodine using lithiation/borylation–protodeboronation methodology

The synthesis of the pharmaceutical (R)-tolterodine is reported using lithiation/borylation–protodeboronation of a homoallyl carbamate as the key step. This step was tested with two permutations: an electron-neutral aryl Li-carbamate reacting with an electron-rich boronic ester and an electron-rich...

Full description

Saved in:
Bibliographic Details
Main Authors: Roesner, Stefan, Aggarwal, Varinder K.
Format: Artigo
Language:Inglês
Published: 2012
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC3672952/
https://ncbi.nlm.nih.gov/pubmed/23750041
Tags: Add Tag
No Tags, Be the first to tag this record!