Enantioselective Copper‐Catalyzed Borylative Cyclization for the Synthesis of Quinazolinones

Quinazolinones are common substructures in molecules of medicinal importance. We report an enantioselective copper‐catalyzed borylative cyclization for the assembly of privileged pyrroloquinazolinone motifs. The reaction proceeds with high enantio‐ and diastereocontrol, and can deliver products cont...

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Detalhes bibliográficos
Publicado no:Angew Chem Int Ed Engl
Main Authors: Dherbassy, Quentin, Manna, Srimanta, Shi, Chunling, Prasitwatcharakorn, Watcharapon, Crisenza, Giacomo E. M., Perry, Gregory J. P., Procter, David J.
Formato: Artigo
Idioma:Inglês
Publicado em: John Wiley and Sons Inc. 2021
Assuntos:
Communications
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC8252434/
https://ncbi.nlm.nih.gov/pubmed/33847459
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.202103259
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