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Molecular Mechanism of β-Arrestin-Biased Agonism at Seven-Transmembrane Receptors

The concept of biased agonism has recently come to the fore with the realization that seven-transmembrane receptors (7TMRs, also known as G protein–coupled receptors, or GPCRs) activate complex signaling networks and can adopt multiple active conformations upon agonist binding. As a consequence, the...

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Autors principals: Reiter, Eric, Ahn, Seungkirl, Shukla, Arun K., Lefkowitz, Robert J.
Format: Artigo
Idioma:Inglês
Publicat: 2011
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3628752/
https://ncbi.nlm.nih.gov/pubmed/21942629
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1146/annurev.pharmtox.010909.105800
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