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Metabolism and Pharmacokinetics of the Anti-Tuberculosis Drug Ethionamide in a Flavin-Containing Monooxygenase Null Mouse

Multiple drug resistance (MDR) in Mycobacterium tuberculosis (mTB), the causative agent for tuberculosis (TB), has led to increased use of second-line drugs, including ethionamide (ETA). ETA is a prodrug bioactivated by mycobacterial and mammalian flavin-containing monooxygenases (FMOs). FMO2 is the...

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Bibliografski detalji
Glavni autori: Palmer, Amy L., Leykam, Virginia L., Larkin, Andrew, Krueger, Sharon K., Phillips, Ian R., Shephard, Elizabeth A., Williams, David E.
Format: Artigo
Jezik:Inglês
Izdano: MDPI 2012
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3621790/
https://ncbi.nlm.nih.gov/pubmed/23580869
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ph5111147
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