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Human Flavin-Containing Monooxygenase 2.1 Catalyzes Oxygenation of the Antitubercular Drugs Thiacetazone and Ethionamide

The second-line antitubercular drugs thiacetazone (TAZ) and ethionamide (ETA) are bioactivated by the mycobacterial enzyme EtaA. We report here that human flavin-containing monooxygenase 2.1 (FMO2.1), which is expressed predominantly in the lung, catalyzes oxygenation of TAZ. The metabolites generat...

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Detalhes bibliográficos
Main Authors: Francois, Asvi A., Nishida, Clinton R., de Montellano, Paul R. Ortiz, Phillips, Ian R., Shephard, Elizabeth A.
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Pharmacology and Experimental Therapeutics 2009
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2683658/
https://ncbi.nlm.nih.gov/pubmed/18948378
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.108.024158
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