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Direct and selective small-molecule activation of proapoptotic BAX

BCL-2 family proteins are key regulators of the apoptotic pathway. Antiapoptotic members sequester the BCL-2 homology 3 (BH3) death domains of proapoptotic members such as BAX to maintain cell survival. The antiapoptotic BH3-binding groove has been successfully targeted to reactivate apoptosis in ca...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Gavathiotis, Evripidis, Reyna, Denis E, Bellairs, Joseph A, Leshchiner, Elizaveta S, Walensky, Loren D
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2012
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3617124/
https://ncbi.nlm.nih.gov/pubmed/22634637
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nchembio.995
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