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Thrombospondin-1 expression in melanoma is blocked by methylation and targeted reversal by 5-Aza-deoxycytidine suppresses angiogenesis

BACKGROUND: Reversibility of aberrant methylation via pharmacological means is an attractive target for therapies through epigenetic reprogramming. To establish that pharmacologic reversal of methylation could result in functional inhibition of angiogenesis, we undertook in vitro and in vivo studies...

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Autores principales: Lindner, Daniel J., Wu, Yan, Haney, Rebecca, Jacobs, Barbara S., Fruehauf, John P., Tuthill, Ralph, Borden, Ernest C.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2012
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3615071/
https://ncbi.nlm.nih.gov/pubmed/23202046
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.matbio.2012.11.010
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