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Comparative in vitro metabolism of phospho-tyrosol-indomethacin by mice, rats and humans

Phospho-tyrosol-indomethacin (PTI; MPI 621), a novel anti-cancer agent, is more potent and safer than conventional indomethacin. Here, we show that PTI was extensively metabolized in vitro and in vivo. PTI was rapidly hydrolyzed by carboxylesterases to generate indomethacin as its major metabolite i...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Xie, Gang, Zhou, Dingying, Cheng, Ka-Wing, Wong, Chi C., Rigas, Basil
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2013
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3604040/
https://ncbi.nlm.nih.gov/pubmed/23399640
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2013.01.031
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