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A structure-activity relationship study on multi-heterocyclic molecules: two linked thiazoles are required for cytotoxic activity

We report the synthesis, cytotoxicity, and phenotypic analysis of oxazole and thiazole containing fragments. Evaluating the optimal size and heterocycle for growth inhibition and apoptosis showed that activity required at least two thiazoles sequentially connected. This is the first detailed compari...

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Bibliographic Details
Main Authors: Kim, Seong Jong, Lin, Chun Chieh, Pan, Chung-Mao, Rananaware, Dimple P., Ramsey, Deborah M., McAlpine, Shelli R.
Format: Artigo
Language:Inglês
Published: 2012
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC3601786/
https://ncbi.nlm.nih.gov/pubmed/23524379
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/C2MD20291C
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