The Potent Human Immunodeficiency Virus Type 1 (HIV-1) Entry Inhibitor HR212 Blocks Formation of the Envelope Glycoprotein gp41 Six-Helix Bundle

Eitemau Tebyg

• N-Substituted Pyrrole Derivatives as Novel Human Immunodeficiency Virus Type 1 Entry Inhibitors That Interfere with the gp41 Six-Helix Bundle Formation and Block Virus Fusion
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  Cyhoeddwyd: (2004)
• Evidence That the Transition of HIV-1 Gp41 into a Six-Helix Bundle, Not the Bundle Configuration, Induces Membrane Fusion
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  Cyhoeddwyd: (2000)
• Resistance to N-peptide fusion inhibitors correlates with thermodynamic stability of the gp41 six-helix bundle but not HIV entry kinetics
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  Cyhoeddwyd: (2014)
• Inhibition of HIV Entry by Targeting the Envelope Transmembrane Subunit gp41
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  Cyhoeddwyd: (2016)
• N-Substituted Pyrrole Derivative 12m Inhibits HIV-1 Entry by Targeting Gp41 of HIV-1 Envelope Glycoprotein
  gan: Qiu, Jiayin, et al.
  Cyhoeddwyd: (2019)