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Current understanding of LRRK2 in Parkinson's disease: biochemical and structural features and inhibitor design

Since leucine-rich repeat kinase 2 (LRRK2) was linked to Parkinson's disease in 2004, kinase activity of LRRK2 has been believed to play a critical role in the pathogenesis of Parkinson's disease. As a result, identification of LRRK2 inhibitors has been a focus for drug discovery. However,...

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Autores principales: Ray, Soumya, Liu, Min
Formato: Artigo
Lenguaje:Inglês
Publicado: 2012
Materias:
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3569718/
https://ncbi.nlm.nih.gov/pubmed/22924508
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.4155/fmc.12.110
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