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Structures of a Na(+)-coupled, substrate-bound MATE multidrug transporter

Multidrug transporters belonging to the multidrug and toxic compound extrusion (MATE) family expel dissimilar lipophilic and cationic drugs across cell membranes by dissipating a preexisting Na(+) or H(+) gradient. Despite its clinical relevance, the transport mechanism of MATE proteins remains poor...

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Autors principals: Lu, Min, Symersky, Jindrich, Radchenko, Martha, Koide, Akiko, Guo, Yi, Nie, Rongxin, Koide, Shohei
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 2013
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3568332/
https://ncbi.nlm.nih.gov/pubmed/23341609
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1219901110
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