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A C-terminally amidated analogue of ShK is a potent and selective blocker of the voltage-gated potassium channel Kv1.3

ShK, a 35-residue peptide from a sea anemone, is a potent blocker of potassium channels. Here we describe a new ShK analogue with an additional C-terminus Lys residue and amide. ShK-K-amide is a potent blocker of Kv1.3 and, in contrast to ShK and ShK-amide, is selective for Kv1.3. To understand this...

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Autori principali: Pennington, Michael W., Rashid, M. Harunur, Tajhya, Rajeev B., Beeton, Christine, Kuyucak, Serdar, Norton, Raymond S.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2012
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3496055/
https://ncbi.nlm.nih.gov/pubmed/23063513
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.febslet.2012.09.038
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