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In Silico and Intuitive Predictions of CYP46A1 Inhibition by Marketed Drugs with Subsequent Enzyme Crystallization in Complex with Fluvoxamine

Cytochrome P450 46A1 (cholesterol 24-hydroxylase) is an important brain enzyme that may be inhibited by structurally distinct pharmaceutical agents both in vitro and in vivo. To identify additional inhibitors of CYP46A1 among U.S. Food and Drug Administration-approved therapeutic agents, we used in...

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Autors principals: Mast, Natalia, Linger, Marlin, Clark, Matthew, Wiseman, Jeffrey, Stout, C. David, Pikuleva, Irina A.
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2012
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3477228/
https://ncbi.nlm.nih.gov/pubmed/22859721
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.112.080424
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