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Antifungal Azoles: Structural Insights into Undesired Tight Binding to Cholesterol-Metabolizing CYP46A1

Although there are currently three generations of antifungal azoles on the market, even the third-generation agents show undesirable interactions with human cytochrome P450 (P450) enzymes. CYP46A1 is a cholesterol-metabolizing P450 in the brain that tightly binds a number of structurally distinct az...

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Autors principals: Mast, Natalia, Zheng, Wenchao, Stout, C. David, Pikuleva, Irina A.
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2013
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3684827/
https://ncbi.nlm.nih.gov/pubmed/23604141
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.113.085902
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