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Microsome biocolloids for rapid drug metabolism and inhibition assessment by LC-MS

Rat liver microsomes attached to nanoparticles were used for LC-MS studies of CYP3A and 2E1 enzymes in metabolism of N-nitroso compounds. Using these biocolloids, turnover rates were measured within 2 min. Inhibitor IC(50) values for ketoconazole (KET) and 4-methylpyrazole (4-MEP) were estimated.

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Bibliografiske detaljer
Main Authors: Bajrami, Besnik, Krishnan, Sadagopan, Rusling, James F.
Format: Artigo
Sprog:Inglês
Udgivet: 2008
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3473178/
https://ncbi.nlm.nih.gov/pubmed/19356087
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