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Dynamics of target-mediated drug disposition: characteristic profiles and parameter identification

In this paper we present a mathematical analysis of the basic model for target mediated drug disposition (TMDD). Assuming high affinity of ligand to target, we give a qualitative characterisation of ligand versus time graphs for different dosing regimes and derive accurate analytic approximations of...

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Autors principals: Peletier, Lambertus A., Gabrielsson, Johan
Format: Artigo
Idioma:Inglês
Publicat: Springer US 2012
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3446204/
https://ncbi.nlm.nih.gov/pubmed/22851162
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10928-012-9260-6
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