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Membrane physical properties influence transmembrane helix formation

The pHLIP peptide has three states: (I) soluble in aqueous buffer, (II) bound to the bilayer surface at neutral pH, and (III) inserted as a transmembrane (TM) helix at acidic pH. The membrane insertion of pHLIP at low pH can be used to target the acidic tissues characteristic of different diseases,...

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Autori principali: Barrera, Francisco N., Fendos, Justin, Engelman, Donald M.
Natura: Artigo
Lingua:Inglês
Pubblicazione: National Academy of Sciences 2012
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3437862/
https://ncbi.nlm.nih.gov/pubmed/22908237
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1212665109
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