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Mechanism-Based Inactivation of Cytochrome P450 2B6 by Methadone through Destruction of Prosthetic Heme

Methadone is a μ-opioid receptor agonist widely used in the treatment of narcotic addiction and chronic pain conditions. Methadone is metabolized predominantly in the liver by cytochromes P450 to its pharmacologically inactive primary metabolite 2-ethylidene-1,5-dimethyl-3,3-diphenylpyrrolidine. Ini...

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Bibliografiska uppgifter
Huvudupphovsmän: Amunugama, Hemali T., Zhang, Haoming, Hollenberg, Paul F.
Materialtyp: Artigo
Språk:Inglês
Publicerad: The American Society for Pharmacology and Experimental Therapeutics 2012
Ämnen:
Länkar:https://ncbi.nlm.nih.gov/pmc/articles/PMC3422545/
https://ncbi.nlm.nih.gov/pubmed/22685215
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.112.045971
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