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Assay Format as a Critical Success Factor for Identification of Novel Inhibitor Chemotypes of Tissue-Nonspecific Alkaline Phosphatase from High-Throughput Screening

The tissue-nonspecific alkaline phosphatase (TNAP) isozyme is centrally involved in the control of normal skeletal mineralization and pathophysiological abnormalities that lead to disease states such as hypophosphatasia, osteoarthritis, ankylosis and vascular calcification. TNAP acts in concert with...

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Autors principals: Chung, Thomas D.Y., Sergienko, Eduard, Millán, José Luis
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2010
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3392958/
https://ncbi.nlm.nih.gov/pubmed/20657462
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules15053010
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