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8-(3-Isothiocyanatostyryl)caffeine Is a Selective, Irreversible Inhibitor of Striatal A(2)-Adenosine Receptors

8-(3-Isothiocyanatostyryl)caffeine (ISC) was synthesized and shown to inhibit selectively the binding of [(3)H]CGS 21680 (an A(2a)-selective agonist) at adenosine receptors in striatal membranes. The K(i) value at A(2a)-receptors was found to be 110 nM (rat), with selectivity ratios for A(2a) versus...

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Hlavní autoři: Ji, Xiao-duo, Gallo-Rodriguez, Carola, Jacobson, Kenneth A.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2004
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3392128/
https://ncbi.nlm.nih.gov/pubmed/22787287
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/ddr.430290407
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