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8-(3-Chlorostyryl)caffeine (CSC) is a selective A(2)-adenosine antagonist in vitro and in vivo
An adenosine antagonist, 8-(3-chlorostyryl)caffeine (CSC), was shown previously to be 520-fold selective for A(2a)-adenosine receptors in radioligand binding assays in the rat brain. In reversing agonist effects on adenylate cyclase, CSC was 22-fold selective for A(2d) receptors in rat pheochromocy-...
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| Главные авторы: | , , , , , |
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| Формат: | Artigo |
| Язык: | Inglês |
| Опубликовано: |
1993
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| Предметы: | |
| Online-ссылка: | https://ncbi.nlm.nih.gov/pmc/articles/PMC3468328/ https://ncbi.nlm.nih.gov/pubmed/8495727 |
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