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Saquinavir Inhibits the Malaria Parasite's Chloroquine Resistance Transporter

The antiretroviral protease inhibitors (APIs) ritonavir, saquinavir, and lopinavir, used to treat HIV infection, inhibit the growth of Plasmodium falciparum at clinically relevant concentrations. Moreover, it has been reported that these APIs potentiate the activity of chloroquine (CQ) against this...

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Autori principali: Martin, Rowena E., Butterworth, Alice S., Gardiner, Donald L., Kirk, Kiaran, McCarthy, James S., Skinner-Adams, Tina S.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Microbiology 2012
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3346596/
https://ncbi.nlm.nih.gov/pubmed/22354298
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.00166-12
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