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STRUCTURE-GUIDED DRUG DESIGN: CONFERRING SELECTIVITY AMONG NEURONAL NICOTINIC RECEPTOR AND ACETYLCHOLINE BINDING PROTEIN SUBTYPES

Neuronal nicotinic receptors, encoded by nine genes of the alpha and three of the beta type of subunits, and whose gene products assemble in distinct permutations as pentameric molecules, constitute a fertile area for structure-guided drug design. Design strategies are augmented by a wide variety of...

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Библиографические подробности
Главные авторы: Taylor, Palmer, Talley, Todd T., Radic’, Zoran, Hansen, Scott B., Hibbs, Ryan E., Shi, Jian
Формат: Artigo
Язык:Inglês
Опубликовано: 2007
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC3341175/
https://ncbi.nlm.nih.gov/pubmed/17826748
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2007.07.038
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